International Journal of Drug Design & Discovery

hi Guest International Journal of Drug Design and Discovery

Volume 1 Issue 1 , January-March 2010         ISSN: 0975-8275

1

Pathophysiological Mechanisms and Therapeutic Drug Targets for Complex Regional Pain Syndrome– Type I

Jegadeesan Vaigunda Ragavendran and Terence J. Coderre

[FULL ARTICLE]

11

Synthesis and Antitubercular Activity of 5-benzyl-3-phenyl dihydroisoxazoles

Surendra Singh Bishta, Arya Ajay, Sudhir Kumar Sinha, Vinita Chaturvedic and Rama P. Tripathi

[FULL ARTICLE]

19

Synthesis, Anti-Tuberculosis and Antiviral Activity of Novel 2-isonicotinoylhydrazono-5-arylidene-4-thiazolidinones

Esra Tatar, İlkay Küçükgüzel, Ş.Güniz Küçükgüzel, Feyza Yılmaz-Demircan, Erik De Clercq,

Graciela Andrei, Robert Snoeck, Christophe Pannecouque, Fikrettin Şahin, Ömer Faruk Bayrak

[FULL ARTICLE]

33

The Stacking Ability of Daunomycin with Base Pairs of DNA: A Theoretical ab Initio (HF) and MP2 Studies

Bipul Bezbaruah, Murshida Karim, Rajib L Sarma and Chitrani Medhi

[FULL ARTICLE]

41

3D QSAR: Exploring Influence of Parameters of Pyrazoline Analogues on Resistant Strains of Staphylococcus aureus

M. S. Bhatia, K. B. Ingale, P. B. Choudhari, B. E. Zarekar, N. M. Bhatia, A. S. Sherikar.

[FULL ARTICLE]

49

Synthesis of 4-(2-ethylphenyl)-1-substituted[1,2,4] triazoloquinazolin-5(4H)-ones for their H1-Antihistamine Activity

V. Alagarsamy, D. Shankar, V. Raja Solomon, P. Parthiban, and J.C. Hanish Singh

[FULL ARTICLE]

57

Synthesis of 6-fluoro-3-(4-piperidinyl)-1,2-benzisoxazole amino acid Derivatives and Anti-DNA Damaging Activity

S. R. Ranganatha, K. Vinaya, S. Chandrappa, C. S. Ananda Kumar, S. B. Benaka Prasad, D. S. Prasanna, K. S. Rangappa

[FULL ARTICLE]

65

Synthesis, In-vitro Evaluation and Computational Studies of Novel Isatinyl Derivatives for their Activity against HIV-TB Co-Infection

Debjani Banerjee, Perumal Yogeeswari, Pritesh Bhat, Anisha Thomas, Dharmarajan Sriram

[FULL ARTICLE]

81

Investigation of the Structural Requirement for 3, 5-disubstituted 4, 5 dihydroisoxazole analogs against M. Tuberculosis: QSAR Study

Revathi A Gupta1, S.G. Kaskhedikar

[FULL ARTICLE]

93

Design and Synthesis of 2-(5-ethyl-pyridine-2-yl) ethanol Analogs as Potential Microbial Agents

Navin B. Patel, Hemant R. Patel

[FULL ARTICLE]

107

Synthesis and Biological Activities of N’-[4-(substituted benzylideneamino)-3-(2′,4′-dichlorophenoxymethyl)-1,2,4-triazol-5yl)] isonicotinyl hydrazides

Rajesh Hunashala, Pradeepkumar Ronad, Veeresh Maddi, Satyanarayana Darbhamulla and Mohammad Kamdod

[FULL ARTICLE]